SCHEMBL28049042

SCHEMBL28049042

CCc1cccc(NBr)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 1/20 0.53
ALDH1A1 P00352 1/20 0.47
SIGMAR1 Q99720 6/20 0.47
MAPT P10636 3/20 0.47
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2A Q12879 1/20 0.47
GRIN2B Q13224 1/20 0.47
GRIN2C Q14957 1/20 0.47
GRIN3A Q8TCU5 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30012057 1.00 RAPGEF4 (0.53) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL30133177 0.83 GRIN2D (0.50) RAPGEF4SIGMAR1GRIN2DGRIN3BGRIN1
SCHEMBL8896899 0.82 RAPGEF4 (0.67) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL16590399 0.81 RAPGEF4 (0.51) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL3617649 0.80 RAPGEF4 (0.55) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL29015003 0.80 ALDH1A1 (0.44) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL11421191 0.78 HDAC4 (0.54) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL11918975 0.78 RAPGEF4 (0.53) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
SCHEMBL5144284 0.78 RAPGEF4 (0.53) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D
Hydrochloric Acid SCHEMBL2868312 0.78 RAPGEF4 (0.53) RAPGEF4ALDH1A1SIGMAR1MAPTGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164104-A Urea derivatives and their use as fatty-acid binding protein (FABP) inhibitors HOFFMANN LA ROCHE 2015-12-16 CN disclosed