SCHEMBL28049332

SCHEMBL28049332

COc1ccc(COC(=O)[C@H](C)N)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.53
ALDH1A1 P00352 3/20 0.53
IDO1 P14902 2/20 0.52
AGXT P21549 2/20 0.52
HTT P42858 2/20 0.50
LDHA P00338 1/20 0.50
ATM Q13315 1/20 0.49
MAPT P10636 1/20 0.49
NPC1 O15118 1/20 0.49
POLB P06746 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MMP9 P14780 2/20 0.48
MMP1 P03956 1/20 0.48
MMP2 P08253 1/20 0.47
MMP12 P39900 1/20 0.47
FFAR1 O14842 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29748635 0.87 ALDH1A1 (0.50) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL31723295 0.86 TDP1 (0.47) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL4456075 0.86 ALDH1A1 (0.55) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL13169359 0.85 ALDH1A1 (0.49) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL3736036 0.84 ALDH1A1 (0.54) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL23750675 0.84 ALDH1A1 (0.54) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL28888054 0.83 ALDH1A1 (0.50) SLC6A4ALDH1A1IDO1AGXTHTT
SCHEMBL28385330 0.83 ALDH1A1 (0.53) ALDH1A1IDO1AGXTHTTLDHA
SCHEMBL16124532 0.82 RAB9A (0.49) ALDH1A1AGXTMAPTNPC1RAB9A
SCHEMBL8570835 0.82 ALDH1A1 (0.55) ALDH1A1IDO1AGXTHTTLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602841-A New ammonium derivative, their preparation method and the pharmaceutical composition containing them 法国施维雅药厂 2018-09-28 CN disclosed
CN-105263519-A Compositions and methods for treating cancer Univ Virginia Patent Found 2016-01-20 CN disclosed