SCHEMBL28051949

SCHEMBL28051949

COCCNc1ccc(C(N)=O)nc1Br

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 4/20 0.47
ALDH1A1 P00352 4/20 0.41
HPGD P15428 1/20 0.41
HCAR3 P49019 2/20 0.40
NCF1 P14598 2/20 0.40
KDM4E B2RXH2 2/20 0.39
UTS2R Q9UKP6 1/20 0.39
RAB9A P51151 2/20 0.38
MAPT P10636 2/20 0.38
GLA P06280 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NNMT P40261 1/20 0.37
NPC1 O15118 1/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28051783 0.82 KDM4E (0.36) ALDH1A1HPGDKDM4ERAB9AMAPT
SCHEMBL28051777 0.80 MAPT (0.41) ALDH1A1HPGDHCAR3KDM4ERAB9A
SCHEMBL16506185 0.79 PTGER4 (0.46) PTGER4ALDH1A1HCAR3NCF1KDM4E
SCHEMBL28271305 0.75 HCAR3 (0.46) PTGER4ALDH1A1HPGDHCAR3KDM4E
SCHEMBL28051766 0.74 ADRA1D (0.48) PTGER4ALDH1A1HPGDHCAR3KDM4E
SCHEMBL16505728 0.73 PTGER4 (0.40) PTGER4ALDH1A1HCAR3NCF1MAPT
SCHEMBL16517756 0.71 PTGER4 (0.50) PTGER4ALDH1A1HCAR3NCF1KDM4E
SCHEMBL4539617 0.70 KDM4E (0.54) PTGER4ALDH1A1HPGDKDM4ERAB9A
SCHEMBL5591756 0.69 PTGER4 (0.47) PTGER4ALDH1A1HCAR3KDM4ERAB9A
SCHEMBL28051782 0.69 PTGER4 (0.47) PTGER4ALDH1A1HPGDHCAR3NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658639-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed