SCHEMBL28051766

SCHEMBL28051766

COCCNc1nccc(C(N)=O)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
KDR P35968 2/20 0.42
IGF1R P08069 1/20 0.42
FGFR1 P11362 1/20 0.42
KDM4E B2RXH2 1/20 0.42
KDM5A P29375 1/20 0.42
JMJD1C Q15652 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42
HCAR3 P49019 1/20 0.42
KCNH3 Q9ULD8 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
ALOX15 P16050 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476571 0.81 HRH4 (0.52) ADRA1DADRA1AADRA1BKDM4EKDM5A
SCHEMBL9196044 0.77 ADRA1D (0.52) ADRA1DADRA1AADRA1BALDH1A1HSD17B10
SCHEMBL19477216 0.77 MKNK1 (0.50) MKNK1MKNK2KDRKDM4EKCNH3
SCHEMBL28271305 0.75 HCAR3 (0.46) KDM4EHCAR3KCNH3ALDH1A1CYP1A2
SCHEMBL3128728 0.75 KDM4E (0.43) ADRA1DADRA1AADRA1BKDRIGF1R
SCHEMBL91582 0.75 MKNK1 (0.51) MKNK1MKNK2KDRKDM4EKCNH3
SCHEMBL9411677 0.75 DRD2 (0.48) ADRA1DADRA1AADRA1B
SCHEMBL13728173 0.75 OPRM1 (0.40) KDRIGF1RFGFR1KDM4EALDH1A1
SCHEMBL16815659 0.75 MKNK1 (0.48) MKNK1MKNK2KDRKDM4EHCAR3
SCHEMBL28051949 0.74 PTGER4 (0.47) KDM4EHCAR3ALDH1A1UTS2RHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658639-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed