SCHEMBL28052832

SCHEMBL28052832

N#CCc1ccc(F)c(C=O)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.39
ERN1 O75460 3/20 0.35
CDK1 P06493 1/20 0.35
FFAR1 O14842 2/20 0.35
FFAR4 Q5NUL3 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
MMP3 P08254 1/20 0.33
PTPRC P08575 1/20 0.33
PTPN1 P18031 1/20 0.33
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556642 0.86 ENPP2 (0.39) ENPP2ERN1CDK1FFAR1FFAR4
SCHEMBL663531 0.79 ENPP2 (0.39) ENPP2ERN1CDK1FFAR1KDM4E
SCHEMBL30694822 0.79 ENPP2 (0.39) ENPP2ERN1CDK1FFAR1KDM4E
SCHEMBL1303380 0.79 CDK1 (0.59) ENPP2ERN1CDK1MMP3
SCHEMBL435376 0.77 HTT (0.41) ENPP2FFAR1FFAR4CYP11B1CYP11B2
SCHEMBL25457596 0.76 LOXL2 (0.41) ERN1CDK1
SCHEMBL12703942 0.76 CYP4F2 (0.46) ENPP2ERN1CDK1
SCHEMBL3854721 0.76 LMNA (0.38) ERN1CDK1NPC1LMNAMAPT
SCHEMBL17149263 0.76 IDO1 (0.41) ERN1CDK1TDP1
SCHEMBL7593948 0.75 TUBB1 (0.47) ERN1KDM4ETDP1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105541769-A Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2016-05-04 CN disclosed
CN-103664637-B Be used for the treatment of ophthalmic diseases and disorderly alkynyl phenyl derivative compounds ACUCELA INC. (US) 2016-02-03 CN disclosed