SCHEMBL28052843

SCHEMBL28052843

COc1ccc(C(=C=O)CC#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA1 P00915 5/20 0.44
CA2 P00918 5/20 0.44
GSK3B P49841 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL135620 0.79 HDAC3 (0.59) CES2CES1NPC1RAB9ALMNA
SCHEMBL28564717 0.77 CES2 (0.45) CES2CES1LMNAMAPTCA1
SCHEMBL28561506 0.77 CES2 (0.45) CES2CES1NPC1LMNAMAPT
SCHEMBL290340 0.76 CES2 (0.46) CES2CES1MEN1MAPTHPGD
SCHEMBL27804569 0.76 CYP19A1 (0.44) CES2CES1MEN1POLBMAPT
Hydrochloric Acid SCHEMBL19379612 0.72 PLK1 (0.45) CES2CES1NPC1RAB9ALMNA
SCHEMBL22767089 0.70 CA1 (0.58) CES2CES1NPC1RAB9AMEN1
SCHEMBL4446152 0.70 NPC1 (0.42) CES2CES1NPC1RAB9ALMNA
SCHEMBL14161830 0.70 CA1 (0.59) CES2CES1RAB9AMEN1LMNA
SCHEMBL6379810 0.69 HDAC3 (0.61) CES2CES1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646358-B A kind of synthetic method of 3 amino 5 (4 anisyl) pyrazoles 苏州艾缇克药物化学有限公司 2018-03-09 CN claimed
CN-105646358-A Synthesizing method of 3-amino-5-(4-methoxyphenyl) pyrazole 苏州艾缇克药物化学有限公司 2016-06-08 CN claimed
CN-105254564-A Synthesis method of 2-methyl-3,4-binitro-5-(methoxyphenyl) pyrazole DING YUQIN 2016-01-20 CN claimed
CN-107739350-B Method for synthesizing 2-aminothiazole derivative 天津大学 2020-12-22 CN disclosed
CN-105646358-B A kind of synthetic method of 3 amino 5 (4 anisyl) pyrazoles 苏州艾缇克药物化学有限公司 2018-03-09 CN disclosed
CN-107739350-A A kind of method for synthesizing 2 aminothiazole derivs 天津大学 2018-02-27 CN disclosed
CN-105646358-A Synthesizing method of 3-amino-5-(4-methoxyphenyl) pyrazole 苏州艾缇克药物化学有限公司 2016-06-08 CN disclosed
CN-105646358-A Synthesizing method of 3-amino-5-(4-methoxyphenyl) pyrazole 苏州艾缇克药物化学有限公司 2016-06-08 CN disclosed
CN-105254564-A Synthesis method of 2-methyl-3,4-binitro-5-(methoxyphenyl) pyrazole DING YUQIN 2016-01-20 CN disclosed