SCHEMBL28053289

SCHEMBL28053289

NC(=O)c1cccc(C=Cc2ccccc2)c1I

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.50
TRPA1 O75762 1/20 0.44
MAPT P10636 5/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
HPGD P15428 2/20 0.44
SIGMAR1 Q99720 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
NFE2L2 Q16236 1/20 0.41
CAPN1 P07384 1/20 0.40
PARP1 P09874 1/20 0.40
BCAT2 O15382 1/20 0.40
BCHE P06276 1/20 0.39
CYP2C19 P33261 1/20 0.39
HDAC3 O15379 1/20 0.39
TNKS O95271 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3639133 0.84 SIRT2 (0.57) SIRT2TRPA1MAPTALDH1A1KDM4E
SCHEMBL2037764 0.84 SIRT2 (0.57) SIRT2TRPA1MAPTALDH1A1KDM4E
SCHEMBL31678976 0.84 SIRT2 (0.57) SIRT2TRPA1MAPTALDH1A1KDM4E
SCHEMBL1415253 0.82 SIRT2 (0.51) SIRT2TRPA1MAPTALDH1A1KDM4E
SCHEMBL1415250 0.74 ALDH1A1 (0.54) SIRT2MAPTALDH1A1KDM4ELMNA
SCHEMBL27486058 0.74 KDM4E (0.52) MAPTALDH1A1KDM4EHPGDSIRT1
SCHEMBL10454313 0.73 NFE2L2 (0.50) TRPA1SIGMAR1NFE2L2
SCHEMBL28410501 0.73 NFE2L2 (0.50) TRPA1SIGMAR1NFE2L2
SCHEMBL2291774 0.73 GRIK1 (0.58) TRPA1MAPTALDH1A1LMNANFE2L2
SCHEMBL29542528 0.73 GRIK1 (0.58) TRPA1MAPTALDH1A1LMNANFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294597-A Benzothiazine derivative, and synthetic method and application thereof UNIV EAST CHINA NORMAL 2016-02-03 CN claimed
CN-105294597-A Benzothiazine derivative, and synthetic method and application thereof UNIV EAST CHINA NORMAL 2016-02-03 CN disclosed