SCHEMBL28053290

SCHEMBL28053290

Cc1ccc(Cc2cccc(C(N)=O)c2I)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
MAPK8 P45983 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
GAA P10253 2/20 0.39
USP2 O75604 1/20 0.39
PARP1 P09874 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MAPT P10636 1/20 0.38
AHR P35869 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SRD5A2 P31213 1/20 0.38
PARP10 Q53GL7 1/20 0.38
HSP90AA1 P07900 1/20 0.38
PLA2G10 O15496 1/20 0.38
PLA2G2A P14555 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30100451 0.85 TSHR (0.51) TSHRMAPK8SIRT2ALDH1A1KDM4E
SCHEMBL28185434 0.85 PLA2G2A (0.49) TSHRSIRT2PARP1PLA2G10PLA2G2A
SCHEMBL4182429 0.84 ALDH1A1 (0.45) TSHRMAPK8SIRT2ALDH1A1KDM4E
SCHEMBL27913154 0.80 MAPK8 (0.43) MAPK8SIRT2ALDH1A1KDM4EHPGD
SCHEMBL30029537 0.77 RPS6KB1 (0.43) MAPK8SIRT2PARP1PARP10
SCHEMBL4523553 0.76 MYC (0.48) TSHRALDH1A1KDM4EHPGDGAA
SCHEMBL10727676 0.75 TSHR (0.54) TSHRALDH1A1KDM4EHPGDMAPT
SCHEMBL4908158 0.73 TSHR (0.72) TSHRALDH1A1NPC1RAB9ASMN1; SMN2
Diethylamine SCHEMBL8601287 0.73 PARP1 (0.41) TSHRMAPK8ALDH1A1KDM4EHPGD
SCHEMBL4848573 0.73 TSHR (0.53) TSHRALDH1A1KDM4EHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294597-A Benzothiazine derivative, and synthetic method and application thereof UNIV EAST CHINA NORMAL 2016-02-03 CN claimed
CN-105294597-A Benzothiazine derivative, and synthetic method and application thereof UNIV EAST CHINA NORMAL 2016-02-03 CN disclosed