SCHEMBL28054286

SCHEMBL28054286

O=CC(=O)c1occ2cccc(Cl)c12

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 2/20 0.33
MAPK1 P28482 2/20 0.32
MCL1 Q07820 1/20 0.31
TERT O14746 1/20 0.31
POLB P06746 1/20 0.30
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23044803 0.82 ALDH1A1 (0.33) ALDH1A1TDP1MAPK1
SCHEMBL27577308 0.82 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ATSHRKDM4E
SCHEMBL28063966 0.81 JAK2 (0.33) ALDH1A1TDP1MAPK1
SCHEMBL23044788 0.81 CES2 (0.33) ALDH1A1MEN1KMT2ATDP1MAPK1
SCHEMBL27902949 0.81 CYP1A2 (0.33) ALDH1A1KDM4EHSD17B10TDP1MAPK1
SCHEMBL27903018 0.77 ALDH1A1 (0.31) ALDH1A1TDP1MAPK1
SCHEMBL8620985 0.73 ALDH1A1 (0.41) ALDH1A1MEN1KMT2AKDM4EHSD17B10
SCHEMBL28275933 0.71 EDNRA (0.48) ALDH1A1KDM4ETDP1MAPK1
SCHEMBL27903016 0.70
SCHEMBL28824909 0.70 ALDH1A1 (0.31) ALDH1A1TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105481864-A Modulators of 5-HT receptors and methods of use thereof ABBOTT GMBH & CO KG ABBOTT LAB 2016-04-13 CN disclosed
CN-105461589-A Acylamino-substituted fused cyclopentanecarboxylic acid derivatives and their use as pharmaceuticals SANOFI AVENTIS 2016-04-06 CN disclosed
CN-105418450-A ACYLAMINO-SUBSTITUTED FUSED CYCLOPENTANECARBOXYLIC ACID DERIVATIVES AND THEIR USE AS PHARMACEUTICALS SANOFI AVENTIS 2016-03-23 CN disclosed
CN-102083432-B Acylamino-substituted fused cyclopentanecarboxylic acid derivatives and their use as pharmaceuticals SANOFI-AVENTIS (FR) 2016-02-17 CN disclosed
CN-102712643-B Modulators of 5-HT receptors and methods of use thereof ABBVIE (US) 2015-12-16 CN disclosed
CN-102712643-A Modulators of 5-HT receptors and methods of use thereof ABBOTT LAB 2012-10-03 CN disclosed