SCHEMBL28054520

SCHEMBL28054520

COC(=O)CCC1CCNC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 2/20 0.47
GABRA5 P31644 2/20 0.47
GABRB2 P47870 2/20 0.47
SLC6A12 P48065 2/20 0.47
SLC6A11 P48066 2/20 0.47
SLC6A13 Q9NSD5 2/20 0.47
GABRA1 P14867 1/20 0.47
GABRR1 P24046 1/20 0.47
GABRA4 P48169 1/20 0.47
TSHR P16473 2/20 0.41
KMT2A Q03164 1/20 0.41
ROCK2 O75116 1/20 0.37
HTR4 Q13639 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
KLK7 P49862 1/20 0.35
SMYD3 Q9H7B4 2/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31566883 0.98 SLC6A1 (0.46) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL1037020 0.90 KMT2A (0.52) SLC6A1SLC6A11SLC6A13TSHRKMT2A
SCHEMBL380886 0.89 TSHR (0.44) TSHRHTR4ALOX15
Hydrochloric Acid SCHEMBL27859719 0.88 KMT2A (0.51) SLC6A1SLC6A11SLC6A13TSHRKMT2A
Hydrochloric Acid SCHEMBL27418446 0.87 GNAI3 (0.43) TSHRKMT2AHTR4ALOX15
Hydrochloric Acid SCHEMBL382045 0.87 GNAI3 (0.43) TSHRKMT2AHTR4ALOX15
Acetic Acid SCHEMBL7427847 0.84 HTR4 (0.41) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
Hydrochloric Acid SCHEMBL31735305 0.83 TSHR (0.46) TSHRKMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL1410339 0.83 SLC6A1 (0.44) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL12571551 0.81 SLC6A1 (0.60) SLC6A1GABRA5GABRB2SLC6A12SLC6A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103118540-B Pesticide containing 2, 5-diketopiperazine derivative as active ingredient Rural Development Office (KR) 2016-02-17 CN claimed
CN-113135924-B Pyrimidine derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-04-26 CN disclosed
CN-113135924-A Pyrimidine derivatives and their use in medicine 广东东阳光药业有限公司 2021-07-20 CN disclosed
CN-103118540-B Pesticide containing 2, 5-diketopiperazine derivative as active ingredient Rural Development Office (KR) 2016-02-17 CN disclosed