SCHEMBL28055770

SCHEMBL28055770

NC(=O)c1cccc(-c2ccc3ccccc3n2)c1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.55
BCAT2 O15382 1/20 0.51
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
IKBKB O14920 1/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
PTGS2 P35354 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
AR P10275 1/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
GMNN O75496 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257294 0.84 BCAT2 (0.53) PARP1BCAT2NPC1RAB9AIKBKB
SCHEMBL31531876 0.84 BCAT2 (0.53) PARP1BCAT2NPC1RAB9AIKBKB
SCHEMBL15903518 0.80 RAB9A (0.52) PARP1BCAT2NPC1RAB9AIKBKB
SCHEMBL2025737 0.77 BCAT2 (0.71) PARP1BCAT2NPC1RAB9AKEAP1
SCHEMBL5106250 0.76 RAB9A (0.62) NPC1RAB9APTGS2MEN1KMT2A
SCHEMBL8830688 0.76 RAB9A (0.55) PARP1NPC1RAB9APTGS2MEN1
Hydrochloric Acid SCHEMBL27966297 0.76 BCAT2 (0.69) PARP1BCAT2NPC1RAB9AKEAP1
Bromide SCHEMBL20502171 0.75 RAB9A (0.50) NPC1RAB9AHCRTR1PTGS2MEN1
SCHEMBL3800586 0.74 IKBKB (0.39) PARP1BCAT2NPC1RAB9AIKBKB
SCHEMBL28129138 0.74 RAB9A (0.56) NPC1RAB9AHCRTR1PTGS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103664876-B Quinoline derivatives and uses thereof SUZHOU SOUTHEAST PHARMACEUTICALS CO., LTD. (CN) 2016-04-20 CN disclosed