SCHEMBL28056179

SCHEMBL28056179

Nc1c(C(F)(F)F)ccc(Cl)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
IDO1 P14902 2/20 0.37
KDR P35968 1/20 0.37
NPFFR2 Q9Y5X5 3/20 0.36
NPFFR1 Q9GZQ6 2/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
DPP4 P27487 1/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5518466 0.82 POLB (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL27401568 0.80 IDO1 (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10825784 0.78 HTR3E (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7574925 0.78 HTR3E (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL14691286 0.77 IDO1 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL102339 0.77 KIF11 (0.41) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL13990216 0.75 HTR3E (0.41) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL21487292 0.75 NOTUM (0.35) IDO1GLAPOLBGAATSHR
SCHEMBL14553804 0.75 GABRA1 (0.36) GLAPOLBGAATSHRKIF11
SCHEMBL9412157 0.74 CA1 (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431427-B Novel PDE 4 inhibitor 明治制果药业株式会社 2017-12-08 CN disclosed
CN-105431427-A Novel PDE4 inhibitor MEIJI SEIKA PHARMA CO LTD 2016-03-23 CN disclosed