SCHEMBL28056272

SCHEMBL28056272

Nc1c(OC(F)(F)F)ccc(F)c1O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.41
EPHX2 P34913 1/20 0.40
MPL P40238 1/20 0.33
KCNN4 O15554 1/20 0.32
KCNH2 Q12809 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
NOS3 P29474 2/20 0.31
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
IDO1 P14902 1/20 0.31
SLC7A5 Q01650 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
APP P05067 1/20 0.30
SCN9A Q15858 1/20 0.30
CDK2 P24941 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21487604 0.79 PDE2A (0.33) PDE2AEPHX2
SCHEMBL28056275 0.79 GRIN2B (0.36) PDE2AEPHX2SCN9A
SCHEMBL15679418 0.79 PDE2A (0.36) PDE2AEPHX2NOS3NOS1NOS2
SCHEMBL31143077 0.76 LMNA (0.39)
SCHEMBL4218979 0.72 ALB (0.39) PDE2AEPHX2MPLKCNN4SCN9A
SCHEMBL14553824 0.72 PDE2A (0.36) PDE2AEPHX2NOS3NOS1NOS2
SCHEMBL102976 0.71 ERN1 (0.39)
SCHEMBL25371124 0.71 MPL (0.40) MPLAPPSCN9A
SCHEMBL28083133 0.70 MPL (0.45) MPLALOX5APFEN1SCN9A
SCHEMBL102339 0.69 KIF11 (0.41) MPLIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431427-B Novel PDE 4 inhibitor 明治制果药业株式会社 2017-12-08 CN disclosed
CN-105431427-A Novel PDE4 inhibitor MEIJI SEIKA PHARMA CO LTD 2016-03-23 CN disclosed