SCHEMBL28056275

SCHEMBL28056275

Nc1c(OC(F)(F)F)ccc(Cl)c1O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.36
SLC1A5 Q15758 2/20 0.35
SCN9A Q15858 3/20 0.34
KMO O15229 2/20 0.34
NOTUM Q6P988 2/20 0.34
AKR1C2 P52895 1/20 0.34
AKR1C1 Q04828 1/20 0.34
ACLY P53396 1/20 0.34
PDE2A O00408 1/20 0.33
EPHX2 P34913 1/20 0.33
EPHX1 P07099 1/20 0.32
S100A9 P06702 1/20 0.32
CXCR2 P25025 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083345 0.81 GRIN2B (0.35) GRIN2BSLC1A5SCN9AKMONOTUM
SCHEMBL28056272 0.79 PDE2A (0.41) SCN9APDE2AEPHX2
SCHEMBL15679418 0.78 PDE2A (0.36) SCN9APDE2AEPHX2
SCHEMBL21487604 0.78 PDE2A (0.33) SLC1A5PDE2AEPHX2
SCHEMBL29917977 0.76 KMO (0.42) SCN9AKMOAKR1C2AKR1C1EPHX2
SCHEMBL28056270 0.74 PDE2A (0.33) GRIN2BSLC1A5KMOAKR1C2AKR1C1
SCHEMBL29778856 0.73 GRIA1 (0.42) GRIN2B
SCHEMBL21603543 0.73 GRIA1 (0.42) GRIN2B
SCHEMBL28056179 0.71 HTR3E (0.44) NOTUM
SCHEMBL14553824 0.70 PDE2A (0.36) SCN9APDE2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431427-B Novel PDE 4 inhibitor 明治制果药业株式会社 2017-12-08 CN disclosed
CN-105431427-A Novel PDE4 inhibitor MEIJI SEIKA PHARMA CO LTD 2016-03-23 CN disclosed