SCHEMBL28056642

SCHEMBL28056642

CCCCCC(=O)ONC(=O)c1cccc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.46
SMPD1 P17405 3/20 0.44
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TSHR P16473 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
THRB P10828 1/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
NR1H4 Q96RI1 1/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11129975 0.84 NAAA (0.54) ALDH1A1HDAC1HDAC2CES2CES1
SCHEMBL31662634 0.84 GAA (0.56) SMN1; SMN2SMPD1NPSR1TSHRCES2
SCHEMBL15993619 0.83 NAAA (0.56) ALDH1A1HDAC1HDAC2CES2CES1
SCHEMBL15923326 0.76 SMN1; SMN2 (0.69) KDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL9168059 0.76 SMN1; SMN2 (0.69) KDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL9168933 0.76 SMN1; SMN2 (0.69) KDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL9574878 0.76 POLB (0.61) ALDH1A1SMN1; SMN2HDAC1HDAC2CES2
SCHEMBL6258472 0.76 SMN1; SMN2 (0.79) KDM4EALDH1A1SMN1; SMN2TSHRHDAC1
SCHEMBL28466653 0.75 P2RX7 (0.39) KDM4ESMN1; SMN2NPSR1CES2CES1
SCHEMBL28446802 0.74 SMPD1 (0.54) ALDH1A1SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107636007-A Beta hairpin peptide mimics 波利弗尔股份公司 2018-01-26 CN disclosed
CN-107001426-A Beta-hairpin peptidomimetics 波利弗尔股份公司 2017-08-01 CN disclosed
CN-107001425-A Beta hairpin peptide mimics 波利弗尔股份公司 2017-08-01 CN disclosed
CN-102844327-B Template-fixed peptidomimetics with CXCR7 modulatory activity 波利弗尔股份公司 2016-10-26 CN disclosed
CN-105849119-A Beta-hairpin peptidomimetics 波利弗尔股份公司 2016-08-10 CN disclosed
CN-105324390-A Beta-hairpin peptidomimetics POLYPHOR AG 2016-02-10 CN disclosed