SCHEMBL28056804

SCHEMBL28056804

CC1(C(=O)O)C=C(c2cccc(F)c2)C=C(C(=O)O)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
KMO O15229 2/20 0.39
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
GPR35 Q9HC97 1/20 0.38
HCAR2 Q8TDS4 1/20 0.36
DCLRE1B Q9H816 1/20 0.36
PIN1 Q13526 1/20 0.35
CCR2 P41597 1/20 0.35
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PLK4 O00444 1/20 0.34
AURKA O14965 1/20 0.34
DAPK3 O43293 1/20 0.34
CHEK2 O96017 1/20 0.34
CDK1 P06493 1/20 0.34
PIM1 P11309 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27775543 0.85 MCL1 (0.39) SMN1; SMN2RARARARBRARG
SCHEMBL27516241 0.85 CA1 (0.39) CA1CA2HCAR2KDM4EAURKA
SCHEMBL27775508 0.85 HCAR3 (0.36) HCAR2RARARARBRARG
SCHEMBL27371651 0.84 BCL2L1 (0.38) GPR35HCAR2CCR2RARARARB
SCHEMBL28186443 0.82 NCOA1 (0.44) NR4A1NR4A2NR4A3GPR35HCAR2
SCHEMBL27798959 0.81 BUB1 (0.34) KMO
SCHEMBL28798118 0.81 HCAR2 (0.38) HCAR2GSK3BDYRK1A
SCHEMBL27975975 0.80 LIPG (0.33) RARARARBRARG
SCHEMBL27749870 0.79 DHODH (0.34) KDRGSK3AGSK3BDYRK1A
SCHEMBL28185681 0.77 HCAR2 (0.34) CA1CA2GPR35HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103874700-B Pyrazolo [3,4-c ] pyridine compounds and methods of use 霍夫曼-拉罗奇有限公司 2018-03-30 CN claimed
CN-105980387-A Serine/threonine kinase inhibitors 阵列生物制药公司 2016-09-28 CN claimed
CN-103874700-B Pyrazolo [3,4-c ] pyridine compounds and methods of use 霍夫曼-拉罗奇有限公司 2018-03-30 CN disclosed
CN-105517547-A Pyrrolo-pyrrole carbamate and related organic compounds, pharmaceutical compositions, and medical uses thereof ABIDE THERAPEUTICS 2016-04-20 CN disclosed