SCHEMBL28057752

SCHEMBL28057752

Nc1ncnc2[nH]cc(-c3ccncc3)c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.48
NTRK1 P04629 8/20 0.47
LRRK2 Q5S007 5/20 0.47
MAPK1 P28482 3/20 0.46
BRAF P15056 1/20 0.46
TNNI3K Q59H18 1/20 0.46
DYRK1A Q13627 4/20 0.44
PRKD3 O94806 3/20 0.44
MAP4K4 O95819 3/20 0.44
PRKACA P17612 3/20 0.44
CLK2 P49760 3/20 0.44
GSK3A P49840 3/20 0.44
GSK3B P49841 3/20 0.44
CDK5 Q00535 3/20 0.44
MAP4K2 Q12851 3/20 0.44
ROCK1 Q13464 3/20 0.44
TAOK1 Q7L7X3 3/20 0.44
CDK8 P49336 2/20 0.44
MAP2K1 Q02750 2/20 0.44
CAMK2A Q9UQM7 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24710755 0.85 LRRK2 (0.51) RETNTRK1LRRK2MAPK1DYRK1A
SCHEMBL7021288 0.85 LRRK2 (0.63) RETNTRK1LRRK2MAPK1BRAF
SCHEMBL1896766 0.82 STK3 (0.58) RETNTRK1LRRK2MAPK1DYRK1A
SCHEMBL4352960 0.82 LRRK2 (0.58) RETNTRK1LRRK2DYRK1APRKD3
SCHEMBL23917432 0.82 LRRK2 (0.50) RETNTRK1LRRK2MAPK1DYRK1A
SCHEMBL8107167 0.82 FLT3 (0.46) RETNTRK1LRRK2MAPK1DYRK1A
SCHEMBL3787081 0.82 SRC (0.50) RETNTRK1LRRK2BRAFTNNI3K
SCHEMBL8107173 0.81 FLT3 (0.46) RETNTRK1LRRK2MAPK1DYRK1A
SCHEMBL28057753 0.81 LRRK2 (0.62) NTRK1LRRK2MAPK1DYRK1APRKD3
SCHEMBL4350812 0.78 KDR (0.57) NTRK1LRRK2MAPK1BRAFTNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431436-A Pyrrolo [2,3-D ] pyrimidine derivatives, processes for their preparation and their use as kinase inhibitors NERVIANO MEDICAL SCIENCES SRL 2016-03-23 CN disclosed