SCHEMBL28058028

SCHEMBL28058028

O=[SH](=O)OCCCNCC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
EPHX2 P34913 9/20 0.41
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TSHR P16473 1/20 0.39
P2RX7 Q99572 2/20 0.38
HSD17B10 Q99714 1/20 0.36
MAPT P10636 1/20 0.35
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DPP4 P27487 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28058016 0.86 EPHX2 (0.44) MEN1KMT2AEPHX2ALDH1A1NPSR1
SCHEMBL28058013 0.77 EPHX2 (0.41) EPHX2ALDH1A1
SCHEMBL10312482 0.71 GRIN2D (0.54) MEN1KMT2AEPHX2ALDH1A1TSHR
SCHEMBL28222413 0.70 KMT2A (0.61) MEN1KMT2AEPHX2ALDH1A1TSHR
SCHEMBL26687399 0.69 KMT2A (0.64) MEN1KMT2AEPHX2ALDH1A1NPSR1
SCHEMBL26687425 0.69 MEN1 (0.59) MEN1KMT2AEPHX2ALDH1A1TSHR
SCHEMBL918262 0.69 MEN1 (0.51) MEN1KMT2AEPHX2ALDH1A1TSHR
SCHEMBL25475060 0.67 KMT2A (0.49) MEN1KMT2AEPHX2ALDH1A1NPSR1
SCHEMBL9289043 0.67 KMT2A (0.53) MEN1KMT2AEPHX2ALDH1A1NPSR1
SCHEMBL21724708 0.67 EPHX2 (0.50) MEN1KMT2AEPHX2ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101597196-B Improved drug candidate and preparation method thereof JIYAKETA CO., LTD. (CH) 2016-05-04 CN disclosed