SCHEMBL28058839

SCHEMBL28058839

CCCN1CCN(OC(=O)C(C)(C)C)C[C@H]1C

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28058929 1.00 DRD3 (0.31) DRD3ALDH1A1GAA
SCHEMBL28055328 0.88 SIGMAR1 (0.39)
SCHEMBL28776242 0.87 DRD3 (0.30) DRD3
SCHEMBL28289023 0.86 DRD3 (0.37) DRD3
SCHEMBL27742729 0.85 SCN1A (0.30)
SCHEMBL27721977 0.85 SCN1A (0.30)
SCHEMBL27722011 0.85 SCN1A (0.30)
SCHEMBL28055265 0.85 HSD11B1 (0.30)
SCHEMBL28290453 0.83 SCN1A (0.34) DRD3ALDH1A1
SCHEMBL28058918 0.81 PARP1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-A Quinazolinones PARP-1 inhibitor and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2019-08-02 CN disclosed
CN-105461697-A Quinazolinone PARP-1 inhibitors, medicinal composition containing inhibitors, and antitumor use of inhibitors INST MATERIA MEDICA CAMS 2016-04-06 CN disclosed