SCHEMBL28059065

SCHEMBL28059065

CS(=O)(=O)c1ccnc(N2CCNCC2)n1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.52
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
ACHE P22303 3/20 0.45
ROCK2 O75116 5/20 0.43
HSP90AA1 P07900 4/20 0.43
HSP90AB1 P08238 4/20 0.43
HRH3 Q9Y5N1 1/20 0.42
LMNA P02545 1/20 0.41
ROCK1 Q13464 1/20 0.40
HTR6 P50406 1/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28059124 0.84 KDM4E (0.43) KDM4EALDH1A1ACHEHSP90AA1HSP90AB1
SCHEMBL5797268 0.76 ADRB1 (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL31518606 0.76 ADRB1 (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
Hydrochloric Acid SCHEMBL5375047 0.74 KDM4E (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
Hydrochloric Acid SCHEMBL7868157 0.74 KDM4E (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL11113633 0.74 ADRB1 (0.61) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL4501470 0.72 ADRB1 (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL7604060 0.72 ADRB1 (0.64) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL5758330 0.72 ADRB1 (0.59) ADRB1KDM4EALDH1A1ACHEROCK2
SCHEMBL573580 0.72 ADRB1 (0.59) ADRB1KDM4EALDH1A1ACHEROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814051-B Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2018-09-25 CN disclosed
CN-105814051-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814041-A Benzotriazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed