SCHEMBL28059516

SCHEMBL28059516

CCn1c2ccccc2c2cc(S(=O)(=O)Nc3ccc(OC)cc3OC)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.53
MAPT P10636 6/20 0.53
MEN1 O00255 4/20 0.53
ALDH1A1 P00352 7/20 0.52
LMNA P02545 6/20 0.52
KEAP1 Q14145 4/20 0.52
NFE2L2 Q16236 4/20 0.52
MAPK1 P28482 2/20 0.52
RAB9A P51151 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
POLB P06746 1/20 0.52
SQSTM1 Q13501 1/20 0.50
TP53 P04637 1/20 0.49
HTT P42858 2/20 0.48
TSHR P16473 2/20 0.48
PKM P14618 1/20 0.48
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
HCRTR1 O43613 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28051136 0.92 KMT2A (0.58) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL28051054 0.85 MAPT (0.67) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL27651554 0.84 MEN1 (0.53) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL27631130 0.84 ALDH1A1 (0.56) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL23148487 0.81 MAPT (0.61) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL28051140 0.78 MAPT (0.64) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL29643325 0.76 MAPT (0.68) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL15466317 0.76 MAPT (0.68) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL28298684 0.76 KMT2A (0.52) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL28051052 0.76 ALDH1A1 (0.53) KMT2AMAPTMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN claimed
CN-105418487-B Carbazole sulfonamide derivative eutectic and preparation method thereof 山西普德药业有限公司 2018-11-02 CN claimed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN claimed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN claimed
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN disclosed
CN-105418487-B Carbazole sulfonamide derivative eutectic and preparation method thereof 山西普德药业有限公司 2018-11-02 CN disclosed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN disclosed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN disclosed