SCHEMBL28059609

SCHEMBL28059609

Oc1ccc(I)cc1OC(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
APP P05067 13/20 0.47
KCNH2 Q12809 4/20 0.41
TMEM97 Q5BJF2 4/20 0.41
SIGMAR1 Q99720 4/20 0.41
ERN1 O75460 1/20 0.38
TRPV1 Q8NER1 1/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16978292 0.80 KCNH2 (0.42) APPKCNH2TMEM97SIGMAR1ERN1
SCHEMBL8778326 0.79 MAOB (0.54) APPKCNH2TMEM97SIGMAR1EPHX2
SCHEMBL2097133 0.78 APP (0.49) APPKCNH2TMEM97SIGMAR1EPHX2
SCHEMBL14121378 0.78 APP (0.49) APPKCNH2TMEM97SIGMAR1EPHX2
SCHEMBL4849499 0.78 APP (0.49) APPKCNH2TMEM97SIGMAR1
SCHEMBL20309112 0.78 EPHX2 (0.39) KCNH2TMEM97SIGMAR1TRPV1EPHX2
SCHEMBL20309036 0.76 NOTUM (0.37) TRPV1EPHX2
SCHEMBL20309114 0.76 TRPV1 (0.32) TRPV1EPHX2
SCHEMBL213780 0.76 MAOA (0.49) APPKCNH2TMEM97SIGMAR1ERN1
SCHEMBL20309113 0.76 NOTUM (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108440515-A Substituted benzofuranyl and benzoxazole based compound and application thereof 卡尔约药物治疗公司 2018-08-24 CN disclosed
CN-105492437-B Substituted benzofuranyl and benzoxazolyl compounds and uses thereof 卡尔约药物治疗公司 2018-05-11 CN disclosed
CN-105492437-A Substituted benzofuranyl and benzoxazolyl compounds and uses thereof KARYOPHARM THERAPEUTICS INC 2016-04-13 CN disclosed