SCHEMBL28060475

SCHEMBL28060475

COC(=O)NC1CCN(OC(=O)C(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.42
ALDH1A1 P00352 1/20 0.41
EPHX1 P07099 2/20 0.40
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
HSD11B1 P28845 2/20 0.36
CYP2C9 P11712 1/20 0.36
DRD2 P14416 2/20 0.36
EPHX2 P34913 2/20 0.36
NAMPT P43490 1/20 0.36
BTK Q06187 1/20 0.36
KCNA3 P22001 1/20 0.35
GAA P10253 1/20 0.35
CKS1B P61024 1/20 0.34
SKP1 P63208 1/20 0.34
SKP2 Q13309 1/20 0.34
KDM5A P29375 1/20 0.34
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28858884 0.81 ALDH1A1 (0.35) CTSKALDH1A1EPHX1EPHX2
SCHEMBL16418439 0.81 CTSK (0.42) CTSKALDH1A1EPHX1CA1CA2
SCHEMBL28865513 0.79 ALDH1A1 (0.58) ALDH1A1DRD2CKS1BSKP1SKP2
SCHEMBL2016955 0.75 EPHX1 (0.68) CTSKALDH1A1EPHX1CA1CA2
SCHEMBL12482202 0.74 SSTR4 (0.42) ALDH1A1
SCHEMBL16349436 0.74 ALDH1A1 (0.38) ALDH1A1EPHX2GAALMNANPSR1
SCHEMBL18166970 0.74 CHRM2 (0.38) ALDH1A1HSD11B1GAA
SCHEMBL8484816 0.74 CTSK (0.50) CTSKEPHX1CA1CA2HSD11B1
SCHEMBL2050427 0.73
SCHEMBL8464579 0.73 EPHX1 (0.46) ALDH1A1EPHX1EPHX2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105399698-A Aromatic heterocyclic derivatives and applications of aromatic heterocyclic derivatives in medicines GUANGDONG HEC PHARMACEUTICAL 2016-03-16 CN disclosed