SCHEMBL28061540

SCHEMBL28061540

N[C@@H](Cc1cnc(-c2cccs2)[nH]1)C(=O)OC(=O)[C@@H](N)Cc1cnc(-c2cccs2)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.41
ERCC1 P07992 7/20 0.38
FEN1 P39748 7/20 0.38
ERCC4 Q92889 7/20 0.38
NTRK1 P04629 1/20 0.37
PBK Q96KB5 1/20 0.35
GRK6 P43250 1/20 0.34
DGAT1 O75907 1/20 0.34
KMT2A Q03164 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRA6 Q16445 1/20 0.34
DNASE1 P24855 1/20 0.33
HPGDS O60760 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497462 0.88 SLC7A5 (0.43) PDE10AERCC1FEN1ERCC4NTRK1
SCHEMBL28061565 0.88 SLC7A5 (0.43) PDE10AERCC1FEN1ERCC4NTRK1
SCHEMBL25754931 0.67 PIN1 (0.58) ERCC1FEN1ERCC4GRK6KMT2A
SCHEMBL2900702 0.66 KDM4E (0.57) ERCC1FEN1ERCC4KMT2A
SCHEMBL10847030 0.63 CYP3A4 (0.53)
SCHEMBL17269663 0.63 GAA (0.47) PDE10AKMT2A
SCHEMBL163444 0.63 CYP3A4 (0.71) KMT2A
SCHEMBL1537285 0.63 CYP3A4 (0.71) KMT2A
SCHEMBL11159530 0.62 HRH1 (0.45)
Hydrochloric Acid SCHEMBL28331180 0.62 CYP3A4 (0.69) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596915-B The synthetic method of 2-thiolhistidine and analogue TETRAHEDRON (FR) 2016-04-20 CN disclosed