SCHEMBL28061565

SCHEMBL28061565

N[C@H](Cc1cnc(-c2cccs2)[nH]1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.43
CYP3A4 P08684 1/20 0.43
PDE10A Q9Y233 2/20 0.42
NTRK1 P04629 1/20 0.40
ERCC1 P07992 2/20 0.40
FEN1 P39748 2/20 0.40
ERCC4 Q92889 2/20 0.40
PKM P14618 2/20 0.39
ALPI P09923 1/20 0.39
PTGS1 P23219 1/20 0.39
XIAP P98170 1/20 0.39
GRK6 P43250 1/20 0.38
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HPGDS O60760 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
PBK Q96KB5 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497462 1.00 SLC7A5 (0.43) SLC7A5CYP3A4PDE10ANTRK1ERCC1
SCHEMBL28061540 0.88 PDE10A (0.41) PDE10ANTRK1ERCC1FEN1ERCC4
SCHEMBL25754931 0.72 PIN1 (0.58) CYP3A4ERCC1FEN1ERCC4PKM
SCHEMBL13095827 0.71 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL59810 0.71 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL5289317 0.71 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL4854900 0.71 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL59078 0.71 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL22403244 0.71 SLC7A5 (0.50) SLC7A5CYP3A4PKMALPIPTGS1
SCHEMBL8957140 0.70 SLC7A5 (0.54) SLC7A5CYP3A4PKMALPIPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596915-B The synthetic method of 2-thiolhistidine and analogue TETRAHEDRON (FR) 2016-04-20 CN disclosed