SCHEMBL28062255

SCHEMBL28062255

O=C(O)Cc1cncc(C(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 2/20 0.36
GABRB2 P47870 2/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 1/20 0.34
GABRA1 P14867 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
GABRR1 P24046 1/20 0.34
GABRR2 P28476 1/20 0.34
GABRA4 P48169 1/20 0.34
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
PMP22 Q01453 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30
AGBL2 Q5U5Z8 1/20 0.30
EGLN1 Q9GZT9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23538172 0.77 CCR1 (0.31)
SCHEMBL27947650 0.75 ADORA2A (0.42) GABRA5GABRB2HSD17B10KDM4ELMNA
SCHEMBL28062239 0.75 AGBL2 (0.38) GABRA5GABRB2HSD17B10ALDH1A1CYP3A4
SCHEMBL5302445 0.72 GABRA5 (0.39) GABRA5GABRB2HSD17B10ALDH1A1CYP3A4
SCHEMBL27912645 0.72 GABRA5 (0.39) GABRA5GABRB2HSD17B10ALDH1A1CYP3A4
SCHEMBL27808822 0.72 GABRA5 (0.47) GABRA5GABRB2HSD17B10ALDH1A1CYP3A4
SCHEMBL20116537 0.72 GABRA5 (0.39) GABRA5GABRB2HSD17B10ALDH1A1CYP3A4
SCHEMBL16369768 0.72 HCAR2 (0.41) HSD17B10ALDH1A1TSHRKDM4ELMNA
SCHEMBL3293609 0.71 IDH1 (0.37)
SCHEMBL29010079 0.69 LMNA (0.34) GABRA5GABRB2HSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473560-A Therapeutically active compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2016-04-06 CN disclosed