SCHEMBL28062313

SCHEMBL28062313

O=[N+]([O-])c1ccc(-c2ncco2)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.43
KCNH2 Q12809 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
POLB P06746 3/20 0.41
ALDH1A1 P00352 2/20 0.41
PTPRC P08575 3/20 0.40
S100A4 P26447 2/20 0.40
MAPT P10636 5/20 0.40
TDP1 Q9NUW8 3/20 0.40
NPBWR1 P48145 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP3A4 P08684 3/20 0.37
PIK3CG P48736 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MCL1 Q07820 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28056041 0.88 PTPRC (0.44) KCNJ1KCNH2MEN1KMT2APOLB
SCHEMBL8689842 0.82 HSD17B10 (0.49) KCNJ1KCNH2MEN1KMT2APOLB
SCHEMBL1127509 0.82 KCNJ1 (0.43) KCNJ1KCNH2MEN1KMT2APOLB
SCHEMBL31463506 0.82 KCNJ1 (0.43) KCNJ1KCNH2MEN1KMT2APOLB
SCHEMBL3978869 0.79 ALDH1A1 (0.46) KCNJ1KCNH2MEN1KMT2AALDH1A1
SCHEMBL1644779 0.79 HSD17B10 (0.49) KCNJ1KCNH2POLBALDH1A1PTPRC
SCHEMBL4265596 0.79 ALDH1A1 (0.49) KCNJ1KCNH2MEN1KMT2APOLB
SCHEMBL11050883 0.77 PTPRC (0.57) MEN1KMT2APOLBALDH1A1PTPRC
SCHEMBL3888275 0.76 ALDH1A1 (0.49) KCNJ1KCNH2MEN1KMT2AALDH1A1
SCHEMBL28062384 0.76 KCNJ1 (0.39) KCNJ1KCNH2MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105517993-A Aryl amide kinase inhibitors BRISTOL MYERS SQUIBB CO 2016-04-20 CN disclosed