SCHEMBL28063135

SCHEMBL28063135

N#Cc1cc(O)c(-c2cccc3ccccc23)c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.46
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
CYP1A2 P05177 1/20 0.40
ACMSD Q8TDX5 1/20 0.39
SLC22A12 Q96S37 2/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALOX15 P16050 1/20 0.38
XDH P47989 1/20 0.38
ANPEP P15144 1/20 0.37
STK10 O94804 1/20 0.37
SLK Q9H2G2 1/20 0.37
CLK1 P49759 1/20 0.37
DYRK1A Q13627 1/20 0.37
GSK3B P49841 1/20 0.37
ADK P55263 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28388485 0.81 MCL1 (0.46) MCL1CA1CA2SLC22A12NCOA3
SCHEMBL15535538 0.81 MCL1 (0.43) MCL1CA1CA2HSP90AA1HSP90AB1
SCHEMBL9640313 0.80 TRPM4 (0.50) MCL1HSP90AA1HSP90AB1CYP1A2ACMSD
SCHEMBL28384020 0.79 IMPDH2 (0.51) MCL1CA1CA2SLC22A12KDM4E
SCHEMBL13170778 0.78 CA1 (0.55) MCL1CA1CA2KDM4EALOX15
SCHEMBL19435497 0.76 SLC22A12 (0.54) CA1CA2HSP90AA1HSP90AB1CYP1A2
SCHEMBL29110490 0.76 MCL1 (0.49) MCL1CA1CA2KDM4EALOX15
SCHEMBL20594987 0.75 MCL1 (0.56) MCL1CA1CA2CYP1A2ACMSD
SCHEMBL29039496 0.75 CA1 (0.50) MCL1CA1CA2HSP90AA1HSP90AB1
SCHEMBL20561064 0.74 MCL1 (0.58) MCL1CA1CA2CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107108478-B URAT1 inhibitors 日本化学药品株式会社 2020-04-24 CN disclosed
CN-105418662-A Preparation and application of cysteine fluorescent probe compound based on BODIPY UNIV JINAN 2016-03-23 CN disclosed