SCHEMBL2806348

SCHEMBL2806348

CCc1cccc(CNc2ncnc3[nH]cnc23)c1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.43
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CA1 P00915 5/20 0.40
CA2 P00918 5/20 0.40
CA7 P43166 5/20 0.40
CA13 Q8N1Q1 5/20 0.40
EGFR P00533 2/20 0.39
PTK2 Q05397 2/20 0.39
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
LMNA P02545 1/20 0.37
ALOX15 P16050 1/20 0.37
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
SLC29A1 Q99808 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2803790 0.90 KMT2A (0.45) HTTNPC1ALDH1A1CA1CA2
SCHEMBL2806350 0.83 LMNA (0.58) HTTNPC1PTK2KMT2ATP53
SCHEMBL4916438 0.82 EGFR (0.56) HTTALDH1A1CA1CA2CA7
SCHEMBL2807686 0.82 TSHR (0.41) HTTEGFRPTK2TP53TSHR
SCHEMBL2805437 0.82 GABRA1 (0.44) HTTPTK2TP53TSHRSMN1; SMN2
SCHEMBL4913797 0.82 EGFR (0.48) HTTNPC1ALDH1A1CA1CA2
SCHEMBL2803307 0.77 CCNB2 (0.42) HTTPTK2TP53TSHRSMN1; SMN2
SCHEMBL2806355 0.76 TDO2 (0.43) HTTNPC1ALDH1A1EGFRTSHR
SCHEMBL4920708 0.76 EGFR (0.42) HTTNPC1ALDH1A1CA1CA2
SCHEMBL2806447 0.76 SLC29A1 (0.51) HTTNPC1ALDH1A1EGFRTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2203451-B1 SUBSTITUTED 6-(ALKYLBENZYLAMINO)PURINE DERIVATIVES FOR USE AS CYTOKININ RECEPTOR ANTAGONISTS AND PREPARATIONS CONTAINING THESE DERIVATIVES UNIV PALACKEHO (CZ) 2014-07-30 EP disclosed
US-20100240537-A1 Substituted 6-(alkylbenzylamino)purine derivatives for use as cytokinin receptor antagonists and preparations containing these derivatives FREIE UNIVERSITAT BERLIN (DE) 2010-09-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240537-A1 Substituted 6-(alkylbenzylamino)purine derivatives for use as cytokinin receptor antagonists and preparations containing these derivatives ADORA2A, P2RY6, P2RY1 HTT 4657/4885NPC1 2741/4885ALDH1A1 1244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.