SCHEMBL28064638

SCHEMBL28064638

Cc1c(C(=O)O)n(C)c2c(F)cccc12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.47
JAK2 O60674 2/20 0.43
BTK Q06187 2/20 0.43
GPR35 Q9HC97 1/20 0.42
TSHR P16473 2/20 0.40
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
RORC P51449 4/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
FABP4 P15090 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALB P02768 1/20 0.36
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064624 0.86 BTK (0.42) MCL1JAK2BTKTSHRKDM4E
SCHEMBL28064659 0.81 MCL1 (0.50) MCL1GPR35TSHRKDM4EL3MBTL1
SCHEMBL23809174 0.78 MCL1 (0.45) MCL1GPR35TSHRKDM4EL3MBTL1
SCHEMBL24756083 0.77 GPR35 (0.45) MCL1GPR35KDM4EL3MBTL1MEN1
SCHEMBL28207997 0.74 MEN1 (0.45) MCL1GPR35TSHRKDM4EL3MBTL1
SCHEMBL28064572 0.74 BTK (0.40) JAK2BTKKDM4ENPC1RAB9A
SCHEMBL30639179 0.73 KDM4E (0.67) MCL1TSHRKDM4EL3MBTL1MEN1
SCHEMBL1092586 0.73 KDM4E (0.67) MCL1TSHRKDM4EL3MBTL1MEN1
SCHEMBL28792536 0.71 HTR2C (0.47) MCL1
SCHEMBL7269233 0.69 PCSK9 (0.52) KDM4EL3MBTL1RORCCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555763-A Indole-carboxamide derivatives HOFFMANN LA ROCHE 2016-05-04 CN disclosed