SCHEMBL28064696

SCHEMBL28064696

CC(=NO)c1cc(F)c(N2CCN(C(=O)OC(C)(C)C)CC2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
MAPT P10636 5/20 0.50
HTT P42858 3/20 0.50
LMNA P02545 2/20 0.45
MAPK1 P28482 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.42
GPR119 Q8TDV5 3/20 0.42
TSHR P16473 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31457120 0.88 ALDH1A1 (0.60) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL8257373 0.88 ALDH1A1 (0.60) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL710108 0.85 ALDH1A1 (0.51) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL21937028 0.82 MAPT (0.51) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL30221908 0.80 SMN1; SMN2 (0.49) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL20521398 0.80 SMN1; SMN2 (0.49) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL28064794 0.80 MAPT (0.47) ALDH1A1MAPTHTTLMNAGPR119
SCHEMBL709255 0.79 MAPT (0.51) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL24125575 0.79 MAPT (0.47) ALDH1A1MAPTHTTLMNAMAPK1
SCHEMBL6128555 0.79 SMARCA2 (0.51) ALDH1A1MAPTHTTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712945-B 2-substituted oxy-5-methylsulfonyl aryl piperazine amide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2020-12-01 CN disclosed
CN-105712945-A 2-Substituted-oxy-5-methylsulfonyl aryl piperazine acidamide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2016-06-29 CN disclosed