SCHEMBL28065520

SCHEMBL28065520

O=c1[nH]ccc2ccnc(-c3ccc(F)cc3)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
RAB9A P51151 2/20 0.40
JAK2 O60674 2/20 0.38
RPS6KA3 P51812 1/20 0.38
MELK Q14680 1/20 0.38
STK24 Q9Y6E0 1/20 0.38
MAPK14 Q16539 5/20 0.38
MAPK11 Q15759 2/20 0.38
MAPK13 O15264 1/20 0.38
RAF1 P04049 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK12 P53778 1/20 0.38
BCHE P06276 1/20 0.38
EGFR P00533 1/20 0.38
CHEK1 O14757 2/20 0.37
CSNK1D P48730 1/20 0.37
MAPK1 P28482 1/20 0.37
GRIA1 P42261 1/20 0.37
GCGR P47871 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17151506 0.77 PDE3B (0.47) PDE3BPDE3ARAB9AMAPK14MAPK11
SCHEMBL4750216 0.77 GRIA1 (0.40) RAB9AJAK2RPS6KA3MELKMAPK14
SCHEMBL14771286 0.70 CHEK1 (0.49) JAK2RPS6KA3MELKSTK24CHEK1
SCHEMBL723954 0.68 AHR (0.47) PDE3BPDE3AMAPK14BCHEEGFR
SCHEMBL4750235 0.68 RAD51 (0.43) RAB9AJAK2RPS6KA3MELKMAPK14
SCHEMBL27418449 0.67 JAK2 (0.41) JAK2RPS6KA3MELKSTK24CHEK1
SCHEMBL28399234 0.67 JAK2 (0.45) JAK2RPS6KA3MELKSTK24CHEK1
SCHEMBL4148219 0.66 PDE3B (0.47) PDE3BPDE3ARAB9AMAPK14MAPK11
SCHEMBL723675 0.64 PIK3CD (0.47) PDE3BPDE3ABCHEGRIA1NPC1
SCHEMBL5983565 0.64 JAK2 (0.41) JAK2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103159757-B The synthetic method of one class 2,7-naphthyridines-1 (2H)-one JIANGSU SIMCERE PHARMACEUTICAL RESEARCH COMPANY LIMITED (CN) 2016-04-20 CN disclosed