SCHEMBL4750216

SCHEMBL4750216

Cc1cc2cc[nH]c(=O)c2c(-c2ccc(F)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADORA2A P29274 3/20 0.40
ADORA1 P30542 3/20 0.40
ADORA2B P29275 2/20 0.40
MAPK14 Q16539 4/20 0.39
MAPK13 O15264 3/20 0.39
MAPK12 P53778 3/20 0.39
MAPK11 Q15759 3/20 0.39
JAK2 O60674 6/20 0.38
CHEK1 O14757 3/20 0.37
IKBKB O14920 1/20 0.37
DAPK3 O43293 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750235 0.77 RAD51 (0.43) ALDH1A1NPC1RAB9AMAPTMAPK14
SCHEMBL28065520 0.77 PDE3B (0.44) GRIA1NPC1RAB9AMAPK14MAPK13
SCHEMBL4243560 0.75 CHEK1 (0.41) ALDH1A1RAB9AKDM4EHPGDADORA2A
SCHEMBL4747721 0.73 KDM4C (0.41) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL12960747 0.72 CHEK1 (0.46) ALDH1A1ADORA2AADORA1JAK2CHEK1
SCHEMBL5815996 0.70 ALDH1A1 (0.37) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL13753079 0.70 JAK2 (0.39) ALDH1A1KDM4EMAPTHPGDADORA2A
SCHEMBL4786704 0.69 AKR1B10 (0.40) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL4751131 0.69 KDM4C (0.38) GRIA1ALDH1A1NPC1RAB9ATP53
SCHEMBL22093860 0.68 JAK2 (0.44) JAK2CHEK1RPS6KA3JAK3MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO disclosed