SCHEMBL28065536

SCHEMBL28065536

Cc1c(Br)c(=O)oc2c(O)c(O)ccc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.79
GAA P10253 5/20 0.79
ALDH1A1 P00352 4/20 0.79
HTT P42858 3/20 0.79
SMN1; SMN2 Q16637 2/20 0.79
CSNK2A1 P68400 1/20 0.79
MAPT P10636 3/20 0.62
MAPK1 P28482 3/20 0.62
POLB P06746 2/20 0.62
BLM P54132 2/20 0.62
LMNA P02545 2/20 0.62
NSD2 O96028 1/20 0.62
HPGD P15428 1/20 0.62
CASP6 P55212 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.62
MCL1 Q07820 2/20 0.56
JAK2 O60674 1/20 0.56
PKM P14618 1/20 0.56
MPI P34949 1/20 0.56
ESR2 Q92731 11/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15285080 0.86 KDM4E (0.61) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL31414410 0.86 KDM4E (0.61) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL2555897 0.81 KDM4E (0.70) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL31060326 0.81 KDM4E (0.70) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL10791581 0.80 KDM4E (0.69) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL19236367 0.79 KDM4E (0.79) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL14756048 0.78 KDM4E (0.53) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL13479651 0.77 KDM4E (1.00) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL8745765 0.75 KDM4E (0.65) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL9318993 0.74 PKLR (0.55) KDM4EGAAALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524034-B Preparation, pharmacological action and the application for treating cerebral ischemia of coumarin derivative 北京大学 2018-08-17 CN disclosed
CN-105566269-B Preparation, pharmacological action and the application for treating itch of coumarin derivative 北京大学 2018-07-10 CN disclosed
CN-105566269-A Preparation and pharmacological effects of coumarin derivative and application of coumarin derivative to treatment on pruritus UNIV BEIJING 2016-05-11 CN disclosed
CN-105524034-A Preparation method of coumarin derivative, pharmacological effect of coumarin derivative and use of coumarin derivative in treatment on cerebral ischemia UNIV BEIJING 2016-04-27 CN disclosed