SCHEMBL28066950

SCHEMBL28066950

NC([C]=O)c1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
CYP2A6 P11509 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX5 P09917 1/20 0.37
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
CA2 P00918 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C19 P33261 1/20 0.33
CNR1 P21554 1/20 0.33
DPP4 P27487 1/20 0.33
PYCR1 P32322 1/20 0.32
MAOA P21397 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9665245 0.78 MAPT (0.40) ALDH1A1ALOX15MAPK1CA2MEN1
SCHEMBL29012807 0.76 ESR1 (0.43) CYP1A2ALDH1A1ALOX15CA2MEN1
SCHEMBL11015372 0.76 ADRB2 (0.50) CYP2A6CYP1A2MAPK1MEN1KMT2A
SCHEMBL7867478 0.76 HTR2A (0.39) HTR2ACYP2A6CYP1A2ALOX5ALDH1A1
SCHEMBL11243676 0.76 ESR1 (0.43) CYP1A2ALDH1A1ALOX15CA2MEN1
SCHEMBL23244675 0.76 PYCR1 (0.40) HTR2ACYP2A6CYP1A2ALOX5ALDH1A1
SCHEMBL349497 0.76 ESR1 (0.43) CYP1A2ALDH1A1ALOX15CA2MEN1
SCHEMBL3758015 0.75 DPP4 (0.50) HTR2ADPP4
SCHEMBL1036920 0.75 DPP4 (0.50) HTR2ADPP4
SCHEMBL1036918 0.75 DPP4 (0.50) HTR2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105593230-A Cathepsin cysteine protease inhibitors MERCK SHARP & DOHME 2016-05-18 CN disclosed