SCHEMBL28068183

SCHEMBL28068183

CN(C(=O)OC(C)(C)C)c1ccncc1.NCc1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
CYP17A1 P05093 1/20 0.40
F2 P00734 4/20 0.39
BRD4 O60885 2/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.37
CREBBP Q92793 1/20 0.36
CYP19A1 P11511 1/20 0.36
POLQ O75417 1/20 0.36
LMNA P02545 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
RAB9A P51151 1/20 0.35
NR1H2 P55055 1/20 0.34
MLYCD O95822 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481946 0.88 PAX8 (0.49) PAX8CYP17A1F2BRD4KDM4E
SCHEMBL16856539 0.87 PAX8 (0.49) PAX8LOXL2BRD4KDM4EKMT2A
Potassium SCHEMBL30601778 0.87 PAX8 (0.48) PAX8CYP17A1F2BRD4KDM4E
SCHEMBL14907964 0.79 BRD4 (0.48) PAX8LOXL2BRD4KMT2ACREBBP
SCHEMBL8018111 0.77 PAX8 (0.55) PAX8BRD4KMT2ACREBBPLMNA
SCHEMBL7433171 0.75 MMP13 (0.48) CYP17A1GPR119RAB9ANAMPT
SCHEMBL15948302 0.74 F2 (0.38) PAX8CYP17A1F2KDM4EKMT2A
SCHEMBL12812295 0.74 KDM4E (0.59) LOXL2KDM4EKMT2ALMNARAB9A
SCHEMBL8336083 0.74 CYP17A1 (0.44) CYP17A1CYP19A1LMNAGPR119RAB9A
SCHEMBL7531272 0.73 PAX8 (0.50) PAX8BRD4KMT2ACREBBPLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693730-A Heteroaryl compounds, compositions thereof, and their use as protein kinase inhibitors 西格诺药品有限公司 2016-06-22 CN disclosed