SCHEMBL28069113

SCHEMBL28069113

FC(F)(F)c1cccc(-c2ccc3n[c][nH]c3c2)n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.43
PIM1 P11309 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
IDH1 O75874 6/20 0.39
IDH2 P48735 1/20 0.39
NOTUM Q6P988 1/20 0.37
COMT P21964 1/20 0.36
IRAK4 Q9NWZ3 3/20 0.35
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA3 P34903 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
NT5E P21589 2/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27930461 0.71 TAAR1 (0.43) NT5E
SCHEMBL1246822 0.70 NPBWR1 (0.44)
SCHEMBL27947333 0.70 FGFR1 (0.43)
SCHEMBL31497612 0.69 TGFBR1 (0.44) TGFBR1PIM1PIM3PIM2IDH1
SCHEMBL30627327 0.69 TRPA1 (0.57) TGFBR1PIM1
SCHEMBL27947326 0.68 MAP4K4 (0.39)
SCHEMBL19072795 0.68 MPL (0.54) TGFBR1IDH1IDH2NOTUMCOMT
SCHEMBL30395354 0.68 NOTUM (0.58) IDH1IDH2NOTUMGABRA1GABRG2
SCHEMBL15624402 0.68 NOTUM (0.58) IDH1IDH2NOTUMGABRA1GABRG2
SCHEMBL22337449 0.68 NOTUM (0.47) TGFBR1IDH1IDH2NOTUMGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658645-A Piperidinylbenzimidazole Derivatives as MPGE-1 Inhibitors 诺瓦赛德股份公司 2016-06-08 CN disclosed