SCHEMBL28069134

SCHEMBL28069134

c1cc(-c2c[nH]c3ncccc23)c2cccnc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.66
IKBKE Q14164 3/20 0.64
TBK1 Q9UHD2 3/20 0.64
PDPK1 O15530 3/20 0.56
DYRK1B Q9Y463 1/20 0.55
CDC7 O00311 3/20 0.54
CDK2 P24941 2/20 0.54
MAP4K4 O95819 2/20 0.54
PIM1 P11309 2/20 0.54
PRKACA P17612 2/20 0.54
GSK3B P49841 2/20 0.54
HIPK2 Q9H2X6 2/20 0.54
CLK4 Q9HAZ1 2/20 0.54
ROCK2 O75116 1/20 0.54
IRAK4 Q9NWZ3 1/20 0.54
DYRK1A Q13627 3/20 0.52
NFATC1 O95644 1/20 0.52
CDK9 P50750 2/20 0.50
CDK5 Q00535 2/20 0.50
PLCG1 P19174 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15397138 0.92 TGFBR1 (0.67) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL5618155 0.86 TGFBR1 (0.71) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL15397129 0.83 IKBKE (0.78) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL198641 0.82 MAPT (0.64)
SCHEMBL16572576 0.81 TGFBR1 (0.67) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL15397133 0.80 TGFBR1 (0.69) TGFBR1IKBKETBK1PDPK1CDC7
SCHEMBL12501165 0.80 TGFBR1 (1.00) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL12501144 0.78 IKBKE (1.00) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL12501143 0.78 TGFBR1 (1.00) TGFBR1IKBKETBK1PDPK1DYRK1B
SCHEMBL12501089 0.78 TGFBR1 (0.63) TGFBR1IKBKETBK1PDPK1DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105622605-A Synthesis method of 5-bromo-7-azaindole ITIC MEDCHEM CO LTD 2016-06-01 CN claimed
CN-105622605-A Synthesis method of 5-bromo-7-azaindole ITIC MEDCHEM CO LTD 2016-06-01 CN disclosed