SCHEMBL28069162

SCHEMBL28069162

COC(=O)c1ccc(CCc2ccc(N)cc2C)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
HPGD P15428 2/20 0.56
HSD17B10 Q99714 2/20 0.56
CYP2C9 P11712 1/20 0.56
ALOX15 P16050 1/20 0.56
ALOX12 P18054 1/20 0.56
CYP2C19 P33261 1/20 0.56
CKS1B P61024 1/20 0.56
SKP2 Q13309 1/20 0.56
HIF1A Q16665 1/20 0.56
CCR6 P51684 1/20 0.53
HKDC1 Q2TB90 1/20 0.53
CYP4A11 Q02928 2/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
CYP4F2 P78329 1/20 0.49
MAPT P10636 6/20 0.47
GAA P10253 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12176925 0.83 LOXL2 (0.65) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL28404517 0.83 ALDH1A1 (0.55) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL17529371 0.82 HPGD (0.54) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL16687961 0.80 ALDH1A1 (0.69) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL15358758 0.80 GFER (0.56) ALDH1A1MAOACYP19A1CASP1
SCHEMBL16420936 0.80 CCR6 (0.52) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL3566972 0.78 LOXL2 (0.58) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL70185 0.78 CYP4A11 (0.75) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL16687617 0.78 TDP1 (0.65) TP53ALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL17429664 0.77 CYP4A11 (0.60) TP53ALDH1A1CYP1A2CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316987-B Benzamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-11-17 CN disclosed
CN-105658635-B Thieno naphthenic base or thieno heterocycle analog derivative, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2019-03-08 CN disclosed
CN-105658635-A Thienocycloalkyl or thienoheterocyclic derivatives, preparation method thereof and use thereof in medicine 江苏恒瑞医药股份有限公司 2016-06-08 CN disclosed