SCHEMBL28069422

SCHEMBL28069422

CCOC(=O)CNNc1cccc(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.50
PDCD1 Q15116 1/20 0.49
CD274 Q9NZQ7 1/20 0.49
SETD7 Q8WTS6 1/20 0.47
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 1/20 0.44
MCHR1 Q99705 1/20 0.44
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL696336 0.86 ALDH1A1 (0.52) ALOX15PDCD1CD274SETD7PDK1
SCHEMBL1120518 0.82 GAA (0.53) ALOX15RXFP1ALDH1A1MAPTKMT2A
SCHEMBL1120688 0.80 MAPT (0.59) ALDH1A1MAPTKMT2AMEN1SMN1; SMN2
SCHEMBL11813065 0.78 SETD7 (0.52) ALOX15PDCD1CD274SETD7PDK1
SCHEMBL2489141 0.76 SCN8A (0.51) PDCD1CD274SMN1; SMN2CNR2POLB
SCHEMBL28001927 0.76 PDCD1 (0.46) ALOX15PDCD1CD274SETD7ALDH1A1
SCHEMBL9364693 0.76 GPR35 (0.58) ALOX15PDCD1CD274SETD7PDK1
Benzonitrile SCHEMBL9811793 0.75 SMN1; SMN2 (0.53) PDCD1CD274ALDH1A1MAPTKMT2A
SCHEMBL23354683 0.74 PDCD1 (0.45) ALOX15PDCD1CD274SETD7PDK1
SCHEMBL5886102 0.74 PDCD1 (0.45) ALOX15PDCD1CD274SETD7PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104395312-B The Spirocyclic derivatives of 4,5-dihydro-pyrazolo [3,4-c] pyridin-2-ones, its preparation method and application SICHUAN HAISCO PHARMACEUTICAL CO.,LTD. (CN) 2016-04-27 CN disclosed