SCHEMBL28069484

SCHEMBL28069484

Cc1cccc(NC2CC2)c1C(=O)c1ccc(Br)c(OC(F)F)c1Br

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 4/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.31
PKM P14618 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
HRH1 P35367 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
HTR3A P46098 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5699196 0.74 HTR3E (0.41) KMT2AKDM4EHTR3EHTR3BCHRM4
SCHEMBL28829472 0.71 CYP2C9 (0.41) CCR5TSHRKMT2AKDM4EPKM
SCHEMBL6644570 0.70 ALDH1A1 (0.39) KMT2AKDM4EEPHX2MEN1SMN1; SMN2
SCHEMBL2904257 0.67 MAPT (0.34) KMT2AKDM4EMEN1
SCHEMBL2904253 0.67 MAPT (0.34) KMT2AKDM4EMEN1
SCHEMBL5204690 0.67 MAPT (0.34) KMT2AKDM4EMEN1
SCHEMBL2639019 0.67 ALDH1A1 (0.37) TSHRKMT2AMEN1
SCHEMBL5177356 0.66 MEN1 (0.32) KMT2AMEN1SMN1; SMN2
SCHEMBL6643716 0.66 ERN1 (0.39) TSHRKDM4E
SCHEMBL2898740 0.66 TSHR (0.44) TSHRKMT2AKDM4EMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801482-A Method for preparing 1-cyclopropyl-4-oxo-7-bromine-8-difluoromethoxy-1,4-dihydro-quinoline-3-nonanoic acid-ethyl ester 浙江中欣氟材股份有限公司 2016-07-27 CN claimed
CN-105777631-A Synthesizing method of 1-cyclopropyl-4-oxo-7-bromo-8-difluoromethoxy-1,4-dihydro-quinoline-3-carboxylic acid ethyl ester 浙江中欣氟材股份有限公司 2016-07-20 CN claimed
CN-105801482-A Method for preparing 1-cyclopropyl-4-oxo-7-bromine-8-difluoromethoxy-1,4-dihydro-quinoline-3-nonanoic acid-ethyl ester 浙江中欣氟材股份有限公司 2016-07-27 CN disclosed
CN-105777631-A Synthesizing method of 1-cyclopropyl-4-oxo-7-bromo-8-difluoromethoxy-1,4-dihydro-quinoline-3-carboxylic acid ethyl ester 浙江中欣氟材股份有限公司 2016-07-20 CN disclosed