SCHEMBL5699196

SCHEMBL5699196

FC(F)Oc1c(Br)cccc1NC1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
HRH1 P35367 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
HTR3A P46098 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5699255 0.76 GAA (0.44) KDM4EGAA
SCHEMBL1771083 0.75 MEN1 (0.36) MEN1HTTKMT2A
SCHEMBL28069484 0.74 CCR5 (0.33) HTR3EHTR3BCHRM4CHRM5CHRNB2
SCHEMBL6650054 0.73 EPHX2 (0.34) ROCK2KDM4EGAA
SCHEMBL5699142 0.72 MEN1 (0.31) MEN1HTTKMT2A
SCHEMBL27902978 0.72 HTR3E (0.57) HTR3EHTR3BCHRM4CHRM5CHRNB2
Hydrochloric Acid SCHEMBL28168296 0.70 HTR3E (0.56) HTR3EHTR3BCHRM4CHRM5CHRNB2
SCHEMBL5734957 0.69 HTR3E (0.44) HTR3EHTR3BCHRM4CHRM5CHRNB2
SCHEMBL23043168 0.69 SCN9A (0.36) MEN1HTTKMT2A
Hydrochloric Acid SCHEMBL4103750 0.68 HTR3E (0.40) HTR3EHTR3BCHRM4CHRM5CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362843-B1 N-cyclopropyl-2-difluoromethoxy-3-bromoaniline and intermediate used for production thereof IHARA CHEMICAL IND CO (JP) 2006-06-14 EP disclosed
EP-1362843-B1 N-cyclopropyl-2-difluoromethoxy-3-bromoaniline and intermediate used for production thereof IHARA CHEMICAL IND CO (JP) 2006-06-14 EP disclosed
EP-1031555-B1 DIFLUOROMETHOXYBENZENE DERIVATIVES AND THEIR USE AS INTERMEDIATES IHARA CHEMICAL IND CO (JP) 2005-04-13 EP disclosed
EP-1362843-A2 N-cyclopropyl-2-difluoromethoxy-3-halogenoaniline and intermediate used for production thereof Ihara Chemical Industry Co., Ltd. (JP) 2003-11-19 EP disclosed
US-6316658-B1 QUINOLONE CARBOXYLATE CHEMICAL INTERMEDIATES; MICROBIOCIDES, BACTERICIDES IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2001-11-13 US disclosed
EP-1031555-A1 N-CYCLOPROPYL-2-DIFLUOROMETHOXY-3-HALOGENOANILINES AND INTERMEDIATES FOR THE PREPARATION THEREOF IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2000-08-30 EP disclosed