SCHEMBL28069841

SCHEMBL28069841

O=C(O)c1c(I)cccc1C1c2ccccc2-c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
GAPDH P04406 1/20 0.37
HSPA1A P0DMV8 1/20 0.37
HSPA8 P11142 1/20 0.37
PTPN7 P35236 1/20 0.37
CYP2C9 P11712 1/20 0.37
POLB P06746 1/20 0.36
CYP1A2 P05177 2/20 0.36
TSHR P16473 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28102236 0.85 POLB (0.37) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL9161966 0.82 CA12 (0.57) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL7796836 0.81 CYP2C9 (0.49) CYP2C9CA12CA1CA2CA7
SCHEMBL16771295 0.75 GAPDH (0.41) GAPDHHSPA1AHSPA8PTPN7CA12
SCHEMBL4851263 0.74 CA12 (0.52) CYP1A2TSHRCA12CA1CA2
SCHEMBL5667417 0.72 FOLH1 (0.44) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL28531858 0.71 FOLH1 (0.53) CYP2C9CA12CA1CA2CA7
SCHEMBL6636937 0.71 MYC (0.49) CYP2C9POLBCA12CA1CA2
SCHEMBL3405052 0.70 MMP2 (0.45) HDAC3NCOR2TSHRCA12CA1
SCHEMBL3034481 0.67 ALDH1A1 (0.50) HDAC8TSHRCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105530923-A Aryl ethers and their use PELOTON THERAPEUTICS INC 2016-04-27 CN disclosed