SCHEMBL28069982

SCHEMBL28069982

CC(C[CH]N)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
CTSK P43235 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA12 O43570 1/20 0.31
CA14 Q9ULX7 1/20 0.31
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2D6 P10635 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28705560 0.83 CTSK (0.39) NOS1NOS3NOS2CTSKCA1
SCHEMBL17871166 0.82 CTSK (0.38) NOS1NOS3NOS2CTSKCA1
SCHEMBL9954495 0.80 TSHR (0.35) NOS1NOS3NOS2CTSKCA1
SCHEMBL27733732 0.80 CTSK (0.33) NOS1NOS3NOS2CTSKCA1
SCHEMBL7324930 0.80 CTSK (0.33) NOS1NOS3NOS2CTSKCA1
SCHEMBL16574707 0.80 TSHR (0.35) NOS1NOS3NOS2CTSKCA1
SCHEMBL4901433 0.80 CTSK (0.33) NOS1NOS3NOS2CTSKCA1
SCHEMBL28705561 0.77 CTSK (0.35) NOS1NOS3NOS2CTSKCA1
SCHEMBL28950491 0.77 CTSK (0.35) NOS1NOS3NOS2CTSKCA1
SCHEMBL2687921 0.77 NOS1 (0.38) NOS1NOS3NOS2CTSKCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555781-A Quinazoline derivatives and their use as DNA methyltransferase inhibitors PF MEDICAMENT 2016-05-04 CN disclosed