SCHEMBL28070062

SCHEMBL28070062

CNc1ccc2cc(F)cc(C(=O)OC(C)(C)C)c2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.36
SCN9A Q15858 2/20 0.36
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRA6 Q16445 1/20 0.34
MCHR1 Q99705 2/20 0.33
PARP1 P09874 2/20 0.32
EGFR P00533 1/20 0.32
HCRTR1 O43613 1/20 0.32
ATR Q13535 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.31
NCF1 P14598 1/20 0.31
APP P05067 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4143686 0.72 HRH4 (0.42) PARP1HSD17B10
SCHEMBL28231922 0.72 CYP2C9 (0.34) FPR2SCN9AGABRA1GABRG2GABRB3
SCHEMBL28231924 0.72 HCRTR1 (0.34) FPR2SCN9AGABRA1GABRG2GABRB3
SCHEMBL9722922 0.69 GABRA1 (0.41) FPR2SCN9AGABRA1GABRG2GABRB3
SCHEMBL28825098 0.67 CES2 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL27533980 0.67 ALDH1A1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL20570435 0.66 EGFR (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31757267 0.66 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL29238191 0.66 GABRA1 (0.41) FPR2SCN9AGABRA1GABRG2GABRB3
SCHEMBL8488435 0.66 EGFR (0.41) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105949120-A Four-tooth chelating single quinoline derivative, preparation method thereof and application as metal ion regulator for neurodegenerative disease 广东工业大学 2016-09-21 CN disclosed