SCHEMBL28070394

SCHEMBL28070394

Nc1ncc2cccc(-c3ccc(N4CCOCC4)cc3)c2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.52
DHFR P00374 2/20 0.51
JUN P05412 3/20 0.49
MAPK8 P45983 3/20 0.49
MAPK10 P53779 3/20 0.49
CNR2 P34972 2/20 0.49
PIK3CA P42336 6/20 0.47
FYN P06241 1/20 0.46
ADK P55263 1/20 0.46
MTOR P42345 4/20 0.46
PIK3R1 P27986 3/20 0.46
LCK P06239 1/20 0.45
KIT P10721 1/20 0.45
SRC P12931 1/20 0.45
KDR P35968 1/20 0.45
PIK3CD O00329 2/20 0.45
PIK3CG P48736 1/20 0.45
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28070389 0.86 HRH4 (0.52) DHFRFYNLCKSRCKDR
SCHEMBL28297006 0.83 CNR2 (0.50) TTKDHFRJUNMAPK8MAPK10
SCHEMBL2558872 0.80 DHFR (0.60) DHFRPIK3CAFYNADKMTOR
SCHEMBL16513631 0.76 MAPK10 (0.79) TTKJUNMAPK8MAPK10CDK1
SCHEMBL29847439 0.76 MAPK10 (0.79) TTKJUNMAPK8MAPK10CDK1
SCHEMBL30634004 0.76 ADORA1 (0.49) DHFRLCKKDR
SCHEMBL15228702 0.75 LCK (0.41) DHFRLCKSRCKDRMAPT
SCHEMBL16514799 0.75 JAK2 (0.66) TTKJUNMAPK8MAPK10CDK1
SCHEMBL31114713 0.74 SMN1; SMN2 (0.55) CNR2PIK3CAFYNADKPIK3CG
SCHEMBL28120724 0.74 DHFR (0.52) DHFRLCKSRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105682661-A Certain chemical entities, compositions, and methods 润新生物公司 2016-06-15 CN disclosed