Quinoline

Quinoline

SCHEMBL28071416

O=C(O)c1ccc2ncccc2c1.c1ccc2ncccc2c1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.65
ALOX15 P16050 1/20 0.60
HTT P42858 1/20 0.60
PLK1 P53350 1/20 0.60
DOT1L Q8TEK3 1/20 0.57
ALDH1A1 P00352 6/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
LMNA P02545 1/20 0.57
PABPC1 P11940 1/20 0.56
BCAT1 P54687 1/20 0.56
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
RAB9A P51151 6/20 0.54
MAPT P10636 3/20 0.54
GAA P10253 3/20 0.54
CYP3A4 P08684 1/20 0.54
NPC1 O15118 6/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HPGD P15428 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29489054 0.95 HTT (0.66) MGAMALOX15HTTPLK1DOT1L
SCHEMBL323178 0.95 HTT (0.66) MGAMALOX15HTTPLK1DOT1L
Hydrochloric Acid SCHEMBL998803 0.93 HTT (0.64) MGAMALOX15HTTPLK1DOT1L
Hydrochloric Acid SCHEMBL7309164 0.93 HTT (0.64) MGAMALOX15HTTPLK1DOT1L
Quinoline SCHEMBL28106687 0.90 ALDH1A1 (0.57) MGAMALOX15HTTPLK1ALDH1A1
Terephthalic Acid SCHEMBL27671577 0.90 ALDH1A1 (0.65) MGAMALOX15HTTPLK1DOT1L
Terephthalic Acid SCHEMBL27671578 0.90 ALDH1A1 (0.65) MGAMALOX15HTTPLK1DOT1L
Quinoline SCHEMBL28116161 0.89 MGAM (0.84) MGAMALOX15HTTPLK1DOT1L
Isophthalic Acid SCHEMBL28271214 0.87 ALDH1A1 (0.57) MGAMALOX15HTTPLK1DOT1L
Quinoline SCHEMBL5874527 0.86 ALDH1A1 (0.65) MGAMALOX15HTTPLK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107286182-A Novel oxazolidinone fluoro quinolone derivative and purposes 李靖 2017-10-24 CN claimed
CN-103459382-B For suppressing the heterocyclic compound of PASK 拜奥埃内杰尼克斯公司 2016-06-29 CN claimed
CN-107286182-A Novel oxazolidinone fluoro quinolone derivative and purposes 李靖 2017-10-24 CN disclosed
CN-103764641-B The tricyclic compound of fractional saturation and preparation and application thereof 扎夫根股份有限公司 2016-10-26 CN disclosed
CN-103459382-B For suppressing the heterocyclic compound of PASK 拜奥埃内杰尼克斯公司 2016-06-29 CN disclosed