Itaconate

Itaconate

SCHEMBL28072799

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nearest known ligand 0.52

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Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.32
HCAR2 Q8TDS4 2/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Itaconate SCHEMBL27371070 0.88 ALOX15 (0.56) ALOX15HSD17B10ALDH1A1TSHR
SCHEMBL28016715 0.81 ALOX15 (0.43) ALOX15HSD17B10HCAR2KEAP1NFE2L2
SCHEMBL1428431 0.81 ALDH1A1 (0.48) HSD17B10ALDH1A1TSHRHCAR2KEAP1
SCHEMBL8610770 0.81 ALDH1A1 (0.48) HSD17B10ALDH1A1TSHRHCAR2KEAP1
Itaconate SCHEMBL28200318 0.81 ALOX15 (0.46) ALOX15HSD17B10ALDH1A1TSHRTHRB
Itaconate SCHEMBL20487589 0.80 ALOX15 (0.59) ALOX15HSD17B10ALDH1A1TSHRHCAR2
Dimethyl Maleate SCHEMBL28166828 0.80 ALOX15 (0.57) ALOX15HSD17B10ALDH1A1TSHRHCAR2
Itaconate SCHEMBL15419775 0.80 ALDH1A1 (0.62) ALOX15HSD17B10ALDH1A1TSHRTHRB
Itaconate SCHEMBL29289404 0.79 ALDH1A1 (0.47) ALOX15HSD17B10ALDH1A1TSHRTHRB
Itaconate SCHEMBL8660291 0.79 ALOX15 (0.49) ALOX15HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829577-A Metal surface treating agent 日本帕卡濑精株式会社 2016-08-03 CN disclosed