SCHEMBL28073238

SCHEMBL28073238

O=[N+]([O-])c1ccccc1Nc1ccc(I)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
TDP1 Q9NUW8 2/20 0.51
ALDH1A1 P00352 1/20 0.51
CASP7 P55210 1/20 0.51
EPAS1 Q99814 1/20 0.50
MAPT P10636 5/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
KAT2B Q92831 2/20 0.42
MAP2K1 Q02750 6/20 0.41
MAP2K2 P36507 3/20 0.41
KCNMA1 Q12791 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4940492 0.85 EPAS1 (0.56) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL30615510 0.85 EPAS1 (0.56) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL3571014 0.82 MAPK1 (0.62) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL22583718 0.82 MAPK1 (0.51) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL4379830 0.81 ALDH1A1 (0.58) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL16634860 0.79 HCAR3 (0.63) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL16634858 0.79 HCAR3 (0.63) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL397773 0.79 MAPK1 (0.77) MAPK1L3MBTL1TDP1ALDH1A1CASP7
SCHEMBL3691221 0.77 MAP2K1 (0.48) MAP2K1MAP2K2
SCHEMBL390986 0.77 MAP2K1 (0.58) MAPK1MAP2K1MAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103479604-B N-(virtue amino) sulfamide derivative including polymorph and compositions, its using method and preparation method as mek inhibitor 阿迪生物科学公司 2016-08-10 CN disclosed