SCHEMBL4379830

SCHEMBL4379830

O=[N+]([O-])c1cnccc1Nc1ccc(I)cc1F

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
HTT P42858 2/20 0.58
RAB9A P51151 1/20 0.58
MAPT P10636 1/20 0.53
GAA P10253 1/20 0.48
MAP2K1 Q02750 11/20 0.46
MAP2K2 P36507 1/20 0.46
PRKCZ Q05513 1/20 0.46
IARS2 Q9NSE4 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NUDT1 P36639 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16657375 0.86 ALDH1A1 (0.70) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL18754336 0.84 ALDH1A1 (0.58) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL16634745 0.81 ALDH1A1 (0.54) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL16634742 0.81 ALDH1A1 (0.54) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL16657400 0.81 HTT (0.67) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL28073238 0.81 MAPK1 (0.51) ALDH1A1RAB9AMAPTGAAMAP2K1
SCHEMBL16067604 0.76 ALDH1A1 (0.53) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL985886 0.76 ALDH1A1 (0.63) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL16657372 0.75 ALDH1A1 (0.82) ALDH1A1HTTRAB9AMAPTGAA
SCHEMBL24539455 0.75 MAP2K1 (0.56) MAP2K1MAP2K2PRKCZIARS2NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2012786-A2 PYRIDONE SULFONAMIDES AND PYRIDONE SULFAMIDES AS MEK INHIBITORS Ardea Biosciences, Inc. (US) 2009-01-14 EP disclosed
WO-2007121481-A2 PYRIDONE SULFONAMIDES AND PYRIDONE SULFAMIDES AS MEK INHIBITORS ARDEA BIOSCIENCES, INC. (US) 2007-10-25 WO disclosed